Millipore’s KinaseProfiler service allows researchers to learn about the specificities of their lead compounds or other chemical entities using a panel comprised of hundreds of kinases. Specificity data can help researchers design more potent and targeted compounds to create successful drugs.
KinaseProfiler advantages include: Selection from 283 protein and lipid kinases; single point inhibition data or 10-point IC50curves; choice of 10 µM or KM ATP; gold Standard radiometric protein kinase assays; HTRF PI 3-Kinase assays; and turnaround time of two weeks or less.
Published in Drug Discovery & Development magazine: Vol. 12, No. 4, April, 2009, p.18.